{"id":11906,"date":"2025-07-07T20:27:33","date_gmt":"2025-07-07T12:27:33","guid":{"rendered":"https:\/\/www.shorro.cn\/index.php\/archives\/11906"},"modified":"2025-07-07T20:27:33","modified_gmt":"2025-07-07T12:27:33","slug":"dmapa%e5%9c%a8%e5%8c%bb%e8%8d%af%e4%b8%ad%e9%97%b4%e4%bd%93%e5%90%88%e6%88%90%e4%b8%ad%e7%9a%84%e9%87%8d%e8%a6%81%e6%80%a7%e4%b8%8e%e7%ba%af%e5%ba%a6%e8%a6%81%e6%b1%82","status":"publish","type":"post","link":"https:\/\/www.shorro.cn\/index.php\/archives\/11906","title":{"rendered":"DMAPA\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u7684\u91cd\u8981\u6027\u4e0e\u7eaf\u5ea6\u8981\u6c42"},"content":{"rendered":"
DMAPA\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u7684\u91cd\u8981\u6027\u4e0e\u7eaf\u5ea6\u8981\u6c42<\/strong><\/p>\n\u8bf4\u5230\u5316\u5b66\uff0c\u5f88\u591a\u4eba\u7b2c\u4e00\u53cd\u5e94\u662f\u67af\u71e5\u3001\u590d\u6742\uff0c\u751a\u81f3\u6709\u70b9\u5371\u9669\u3002\u4f46\u5982\u679c\u4f60\u63a5\u89e6\u8fc7\u6709\u673a\u5408\u6210\uff0c\u5c24\u5176\u662f\u533b\u836f\u4e2d\u95f4\u4f53\u7684\u5408\u6210\u9886\u57df\uff0c\u4f60\u4f1a\u53d1\u73b0\uff0c\u8fd9\u91cc\u9762\u5176\u5b9e\u85cf\u7740\u4e00\u95e8\u827a\u672f\u2014\u2014\u7528\u5206\u5b50\u62fc\u56fe\uff0c\u521b\u9020\u51fa\u80fd\u6551\u4eba\u4e8e\u6c34\u706b\u7684\u65b0\u836f\u3002\u800c\u5728\u8fd9\u4e00\u8fc7\u7a0b\u4e2d\uff0c\u6709\u4e00\u79cd\u770b\u4f3c\u4e0d\u8d77\u773c\u5374\u6781\u4e3a\u5173\u952e\u7684\u5316\u5408\u7269\uff0c\u5b83\u5c31\u662f\uff1aN,N-\u4e8c\u7532\u57fa-1,3-\u4e19\u4e8c\u80fa<\/strong>\uff0c\u7b80\u79f0DMAPA<\/strong>\u3002<\/p>\n\u4eca\u5929\uff0c\u6211\u4eec\u5c31\u6765\u804a\u804a\u8fd9\u4e2a\u201c\u5e55\u540e\u82f1\u96c4\u201dDMAPA\uff0c\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u5230\u5e95\u6709\u591a\u91cd\u8981\uff0c\u4ee5\u53ca\u5b83\u7684\u7eaf\u5ea6\u4e3a\u4ec0\u4e48\u4e0d\u80fd\u542b\u7cca\u534a\u5206\u3002<\/p>\n
\n\u4e00\u3001DMAPA\u662f\u4ec0\u4e48\uff1f\u5b83\u4ece\u54ea\u91cc\u6765\uff1f<\/h3>\n
DMAPA\uff0c\u5168\u540d\u662fN,N-\u4e8c\u7532\u57fa-1,3-\u4e19\u4e8c\u80fa<\/strong>\uff0c\u7ed3\u6784\u5f0f\u4e3a CH\u2082CH\u2082NHCH\u2082CH\u2082CH\u2083\uff08\u5f53\u7136\uff0c\u66f4\u51c6\u786e\u70b9\u662f\uff1a(CH\u2083)\u2082NCH\u2082CH\u2082CH\u2082NH\u2082\uff09\uff0c\u662f\u4e00\u79cd\u8102\u80aa\u65cf\u591a\u80fa\u7c7b\u5316\u5408\u7269\u3002\u5b83\u6709\u4e24\u4e2a\u6c28\u57fa\u5b98\u80fd\u56e2\uff0c\u4e00\u4e2a\u4f4d\u4e8e\u94fe\u7aef\uff0c\u4e00\u4e2a\u88ab\u4e24\u4e2a\u7532\u57fa\u53d6\u4ee3\uff0c\u8fd9\u79cd\u7ed3\u6784\u8ba9\u5b83\u5728\u6709\u673a\u5408\u6210\u4e2d\u5177\u6709\u6781\u9ad8\u7684\u7075\u6d3b\u6027\u548c\u53cd\u5e94\u6d3b\u6027\u3002<\/p>\n\u5b83\u901a\u5e38\u901a\u8fc7\u51e0\u79cd\u65b9\u6cd5\u5236\u5907\uff0c\u6bd4\u5982\uff1a<\/p>\n
\n- \u4e59\u8148\u6cd5<\/strong>\uff1a\u7531\u4e59\u8148\u548c\u4e8c\u7f29\u5408\u540e\u8fd8\u539f\u5f97\u5230\uff1b<\/li>\n
- \u4e19\u70ef\u8148\u6cd5<\/strong>\uff1a\u5148\u4e0e\u4e8c\u52a0\u6210\uff0c\u518d\u8fdb\u884c\u6c22\u5316\u8fd8\u539f\uff1b<\/li>\n
- \u5546\u4e1a\u5316\u8def\u7ebf<\/strong>\uff1a\u76ee\u524d\u5927\u591a\u6570\u5de5\u4e1a\u751f\u4ea7\u91c7\u7528\u7684\u662f\u8fde\u7eed\u5316\u5de5\u827a\uff0c\u4ee5\u63d0\u9ad8\u4ea7\u7387\u5e76\u63a7\u5236\u526f\u4ea7\u7269\u3002<\/li>\n<\/ul>\n
\n\n\n\u5236\u5907\u65b9\u6cd5<\/th>\n | \u539f\u6599<\/th>\n | \u53cd\u5e94\u6761\u4ef6<\/th>\n | \u4ea7\u7387<\/th>\n | \u7eaf\u5ea6<\/th>\n<\/tr>\n<\/thead>\n |
\n\n\u4e59\u8148\u6cd5<\/td>\n | \u4e59\u8148\u3001\u4e8c<\/td>\n | \u9ad8\u6e29\u9ad8\u538b\u3001\u50ac\u5316\u5242<\/td>\n | 60%-70%<\/td>\n | \u4e2d\u7b49<\/td>\n<\/tr>\n |
\n\u4e19\u70ef\u8148\u6cd5<\/td>\n | \u4e19\u70ef\u8148\u3001\u4e8c<\/td>\n | \u8fd8\u539f\u52a0\u6c22<\/td>\n | 75%-85%<\/td>\n | \u8f83\u9ad8<\/td>\n<\/tr>\n |
\n\u5de5\u4e1a\u5408\u6210<\/td>\n | \u591a\u6b65\u50ac\u5316<\/td>\n | \u81ea\u52a8\u5316\u8fde\u7eed\u53cd\u5e94<\/td>\n | 90%\u4ee5\u4e0a<\/td>\n | \u9ad8\u7eaf\u5ea6<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n DMAPA\u672c\u8eab\u5916\u89c2\u4e3a\u65e0\u8272\u81f3\u6de1\u9ec4\u8272\u6db2\u4f53\uff0c\u6709\u8f7b\u5fae\u6c28\u5473\uff0c\u6613\u6eb6\u4e8e\u6c34\u548c\u591a\u6570\u6709\u673a\u6eb6\u5242\uff0c\u8fd9\u4f7f\u5f97\u5b83\u5728\u6709\u673a\u5408\u6210\u4e2d\u975e\u5e38\u201c\u597d\u4f7f\u201d\u3002<\/p>\n \n\u4e8c\u3001DMAPA\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u7684\u201c\u95ea\u5149\u65f6\u523b\u201d<\/h3>\n\u533b\u836f\u4e2d\u95f4\u4f53\uff0c\u987e\u540d\u601d\u4e49\uff0c\u662f\u901a\u5f80\u7ec8\u836f\u7269\u7684\u5173\u952e\u4e2d\u95f4\u6b65\u9aa4\u3002\u5f88\u591a\u836f\u7269\u5206\u5b50\u7ed3\u6784\u590d\u6742\uff0c\u76f4\u63a5\u5408\u6210\u56f0\u96be\uff0c\u56e0\u6b64\u9700\u8981\u4e00\u6b65\u6b65\u6784\u5efa\u9aa8\u67b6\uff0c\u800cDMAPA\u6b63\u662f\u5176\u4e2d\u7684\u201c\u7c98\u5408\u5242\u201d\u548c\u201c\u6865\u6881\u201d\u3002<\/p>\n 1. \u4f5c\u4e3a\u4eb2\u6838\u8bd5\u5242\u53c2\u4e0e\u9170\u5316\u53cd\u5e94<\/strong><\/h4>\nDMAPA\u4e2d\u7684\u4ef2\u80fa\u90e8\u5206\u53ef\u4ee5\u4f5c\u4e3a\u826f\u597d\u7684\u4eb2\u6838\u8bd5\u5242\uff0c\u53c2\u4e0e\u591a\u79cd\u9170\u5316\u53cd\u5e94\uff0c\u6bd4\u5982\u4e0e\u9170\u6c2f\u3001\u9178\u9150\u6216\u6d3b\u6027\u916f\u53cd\u5e94\u751f\u6210\u76f8\u5e94\u7684\u9170\u80fa\u3002\u8fd9\u7c7b\u53cd\u5e94\u5e7f\u6cdb\u7528\u4e8e\u5934\u5b62\u7c7b\u6297\u751f\u7d20\u3001\u6297\u6291\u90c1\u836f\u548c\u6297\u9ad8\u8840\u538b\u836f\u7269\u7684\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u3002<\/p>\n \u4f8b\u5982\uff1a<\/p>\n \n\u5728\u67d0\u7c7b\u03b2-\u5185\u9170\u80fa\u7c7b\u6297\u751f\u7d20\u7684\u5408\u6210\u4e2d\uff0cDMAPA\u88ab\u7528\u6765\u6784\u5efa\u5173\u952e\u7684\u4fa7\u94fe\u7ed3\u6784\uff0c\u5e2e\u52a9\u5f15\u5165\u7279\u5b9a\u7684\u5b98\u80fd\u56e2\uff0c\u4ece\u800c\u589e\u5f3a\u836f\u7269\u5bf9\u9776\u70b9\u7684\u9009\u62e9\u6027\u548c\u6297\u83cc\u6d3b\u6027\u3002\n<\/p>\n<\/blockquote>\n 2. \u4f5c\u4e3a\u73af\u5316\u53cd\u5e94\u7684\u6a21\u677f<\/strong><\/h4>\nDMAPA\u5206\u5b50\u4e2d\u542b\u6709\u4e24\u4e2a\u6c28\u57fa\uff0c\u5176\u4e2d\u4e00\u4e2a\u5e26\u53d6\u4ee3\u57fa\uff0c\u53e6\u4e00\u4e2a\u662f\u4f2f\u80fa\uff0c\u8fd9\u79cd\u7ed3\u6784\u975e\u5e38\u9002\u5408\u53d1\u751f\u5206\u5b50\u5185\u73af\u5316\u53cd\u5e94\uff0c\u5c24\u5176\u662f\u5728\u91d1\u5c5e\u50ac\u5316\u4e0b\u5f62\u6210\u4e94\u5143\u6216\u516d\u5143\u6742\u73af\u7ed3\u6784\u3002\u8fd9\u7c7b\u53cd\u5e94\u5e38\u7528\u4e8e\u55b9\u8bfa\u916e\u7c7b\u6297\u83cc\u836f\u548c\u67d0\u4e9b\u6297\u80bf\u7624\u836f\u7269\u7684\u5408\u6210\u8def\u5f84\u4e2d\u3002<\/p>\n 3. \u4f5c\u4e3a\u624b\u6027\u8bf1\u5bfc\u5242\u4f7f\u7528<\/strong><\/h4>\n\u867d\u7136DMAPA\u672c\u8eab\u4e0d\u662f\u624b\u6027\u5206\u5b50\uff0c\u4f46\u5728\u67d0\u4e9b\u4e0d\u5bf9\u79f0\u5408\u6210\u4e2d\uff0c\u5b83\u53ef\u4ee5\u4f5c\u4e3a\u52a9\u50ac\u5316\u5242\u6216\u914d\u4f53\u524d\u4f53\uff0c\u534f\u52a9\u6784\u5efa\u624b\u6027\u4e2d\u5fc3\u3002\u8fd9\u5bf9\u4e8e\u5f00\u53d1\u65b0\u4e00\u4ee3\u7684\u624b\u6027\u836f\u7269\u81f3\u5173\u91cd\u8981\u3002<\/p>\n 4. \u7528\u4e8e\u56fa\u76f8\u5408\u6210\u8f7d\u4f53\u4fee\u9970<\/strong><\/h4>\n\u5728\u73b0\u4ee3\u836f\u7269\u7b5b\u9009\u6280\u672f\u5982\u56fa\u76f8\u5408\u6210\uff08Solid Phase Synthesis\uff09\u4e2d\uff0cDMAPA\u7ecf\u5e38\u88ab\u7528\u6765\u4fee\u9970\u6811\u8102\u8f7d\u4f53\uff0c\u4f7f\u5176\u80fd\u591f\u627f\u8f7d\u66f4\u591a\u79cd\u7c7b\u7684\u53cd\u5e94\uff0c\u63d0\u9ad8\u5408\u6210\u6548\u7387\u548c\u591a\u6837\u6027\u3002<\/p>\n \n\u4e09\u3001DMAPA\u7684\u7eaf\u5ea6\u8981\u6c42\u4e3a\u4f55\u5982\u6b64\u82db\u523b\uff1f<\/h3>\n\u65e2\u7136DMAPA\u8fd9\u4e48\u91cd\u8981\uff0c\u90a3\u5b83\u7684\u8d28\u91cf\u81ea\u7136\u4e0d\u5bb9\u5ffd\u89c6\u3002\u5c24\u5176\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\uff0c\u54ea\u6015\u662f\u4e00\u4e01\u70b9\u6742\u8d28\uff0c\u90fd\u53ef\u80fd\u5f15\u53d1\u8fde\u9501\u53cd\u5e94\uff0c\u5f71\u54cd\u7ec8\u836f\u7269\u7684\u8d28\u91cf\u3001\u5b89\u5168\u6027\u751a\u81f3\u7597\u6548\u3002<\/p>\n 1. \u6742\u8d28\u6765\u6e90\u4e0e\u5f71\u54cd<\/strong><\/h4>\n\u5e38\u89c1\u7684\u6742\u8d28\u5305\u62ec\uff1a<\/p>\n \n- \u672a\u53cd\u5e94\u5b8c\u5168\u7684\u539f\u6599\u6b8b\u7559<\/strong>\uff0c\u5982\u4e8c\u3001\u4e19\u4e8c\u80fa\uff1b<\/li>\n
- \u526f\u4ea7\u7269<\/strong>\uff0c\u5982\u6c27\u5316\u7269\u3001\u805a\u5408\u7269\uff1b<\/li>\n
- \u91cd\u91d1\u5c5e\u6b8b\u7559<\/strong>\uff0c\u5982\u954d\u3001\u94af\u3001\u94dc\u7b49\uff1b<\/li>\n
- \u6c34\u5206\u542b\u91cf\u8fc7\u9ad8<\/strong>\uff0c\u5f71\u54cd\u540e\u7eed\u53cd\u5e94\u7684\u6536\u7387\u548c\u7a33\u5b9a\u6027\u3002<\/li>\n<\/ul>\n
\u8fd9\u4e9b\u6742\u8d28\u5982\u679c\u8d85\u6807\uff0c\u53ef\u80fd\u5bfc\u81f4\uff1a<\/p>\n <\/p>\n
\n- \u672a\u53cd\u5e94\u5b8c\u5168\u7684\u539f\u6599\u6b8b\u7559<\/strong>\uff0c\u5982\u4e8c\u3001\u4e19\u4e8c\u80fa\uff1b<\/li>\n
- \u526f\u4ea7\u7269<\/strong>\uff0c\u5982\u6c27\u5316\u7269\u3001\u805a\u5408\u7269\uff1b<\/li>\n
- \u91cd\u91d1\u5c5e\u6b8b\u7559<\/strong>\uff0c\u5982\u954d\u3001\u94af\u3001\u94dc\u7b49\uff1b<\/li>\n
- \u6c34\u5206\u542b\u91cf\u8fc7\u9ad8<\/strong>\uff0c\u5f71\u54cd\u540e\u7eed\u53cd\u5e94\u7684\u6536\u7387\u548c\u7a33\u5b9a\u6027\u3002<\/li>\n<\/ul>\n
\u8fd9\u4e9b\u6742\u8d28\u5982\u679c\u8d85\u6807\uff0c\u53ef\u80fd\u5bfc\u81f4\uff1a<\/p>\n \n- \u5408\u6210\u5931\u8d25\u6216\u6536\u7387\u964d\u4f4e\uff1b<\/li>\n
- \u836f\u7269\u4e2d\u95f4\u4f53\u4e2d\u6b8b\u7559\u6742\u8d28\u8d85\u6807\uff1b<\/li>\n
- \u7ec8\u836f\u7269\u4e0d\u7b26\u5408GMP\u6807\u51c6\uff1b<\/li>\n
- \u5bf9\u4eba\u4f53\u4ea7\u751f\u6bd2\u526f\u4f5c\u7528\u3002<\/li>\n<\/ul>\n
2. \u884c\u4e1a\u6807\u51c6\u4e0e\u68c0\u6d4b\u6307\u6807<\/strong><\/h4>\n\u4e3a\u4e86\u786e\u4fddDMAPA\u7b26\u5408\u533b\u836f\u7ea7\u6807\u51c6\uff0c\u901a\u5e38\u9700\u8981\u6ee1\u8db3\u4ee5\u4e0b\u53c2\u6570\uff1a<\/p>\n \n\n\n\u68c0\u6d4b\u9879\u76ee<\/th>\n | \u533b\u836f\u7ea7\u6807\u51c6<\/th>\n | \u5de5\u4e1a\u7ea7\u6807\u51c6<\/th>\n<\/tr>\n<\/thead>\n | \n\n\u542b\u91cf<\/td>\n | \u226599.0%<\/td>\n | \u226595.0%<\/td>\n<\/tr>\n | \n\u6c34\u5206<\/td>\n | \u22640.5%<\/td>\n | \u22642.0%<\/td>\n<\/tr>\n | \n\u6b8b\u7559\u6eb6\u5242<\/td>\n | \u7b26\u5408ICH Q3C<\/td>\n | \u4e0d\u4e25\u683c<\/td>\n<\/tr>\n | \n\u91cd\u91d1\u5c5e\uff08Pb\u3001As\uff09<\/td>\n | \u226410 ppm<\/td>\n | \u226450 ppm<\/td>\n<\/tr>\n | \n\u7535\u5bfc\u7387<\/td>\n | \u226410 \u03bcS\/cm<\/td>\n | \u65e0\u660e\u786e\u8981\u6c42<\/td>\n<\/tr>\n | \n\u6c14\u5473\/\u989c\u8272<\/td>\n | \u65e0\u660e\u663e\u523a\u6fc0\u6c14\u5473\uff0c\u900f\u660e\u6216\u5fae\u9ec4<\/td>\n | \u53ef\u7565\u5e26\u5f02\u5473<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n \u6b64\u5916\uff0c\u8fd8\u9700\u505aGC\u6216HPLC\u5206\u6790\u5176\u7eaf\u5ea6\uff0c\u5e76\u5b9a\u671f\u8fdb\u884c\u5fae\u751f\u7269\u9650\u5ea6\u68c0\u67e5\uff0c\u786e\u4fdd\u65e0\u83cc\u6027\u3002<\/p>\n 3. \u7eaf\u5ea6\u4e0e\u6210\u672c\u7684\u535a\u5f08<\/strong><\/h4>\n\u867d\u7136\u6211\u4eec\u5e0c\u671bDMAPA\u8d8a\u7eaf\u8d8a\u597d\uff0c\u4f46\u73b0\u5b9e\u603b\u662f\u8981\u8bb2\u6027\u4ef7\u6bd4\u3002\u5236\u836f\u516c\u53f8\u5f80\u5f80\u4f1a\u6839\u636e\u5177\u4f53\u7528\u9014\u9009\u62e9\u4e0d\u540c\u7ea7\u522b\u7684\u4ea7\u54c1\uff1a<\/p>\n \n- \u9ad8\u7aef\u65b0\u836f\u7814\u53d1\u9636\u6bb5<\/strong>\uff1a\u5fc5\u987b\u4f7f\u7528\u9ad8\u7eaf\u5ea6\u3001\u4f4e\u6742\u8d28\u7684\u533b\u836f\u7ea7DMAPA\uff1b<\/li>\n
- \u4eff\u5236\u836f\u6216\u7c97\u54c1\u5408\u6210\u9636\u6bb5<\/strong>\uff1a\u53ef\u9002\u5f53\u653e\u5bbd\u6807\u51c6\uff0c\u964d\u4f4e\u6210\u672c\uff1b<\/li>\n
- \u4e2d\u95f4\u4f53\u653e\u5927\u8bd5\u9a8c\u9636\u6bb5<\/strong>\uff1a\u9700\u5e73\u8861\u8d28\u91cf\u548c\u4ea7\u91cf\uff0c\u9009\u62e9\u7a33\u5b9a\u4f9b\u5e94\u5546\u3002<\/li>\n<\/ul>\n
\n\u56db\u3001DMAPA\u7684\u5e94\u7528\u6848\u4f8b\u5206\u4eab<\/h3>\n\u4e3a\u4e86\u8ba9\u5927\u5bb6\u66f4\u76f4\u89c2\u5730\u7406\u89e3DMAPA\u7684\u91cd\u8981\u6027\uff0c\u6211\u4eec\u6765\u770b\u51e0\u4e2a\u771f\u5b9e\u5e94\u7528\u6848\u4f8b\u3002<\/p>\n \u6848\u4f8b\u4e00\uff1a\u5934\u5b62\u514b\u809f\u7684\u5408\u6210<\/h4>\n\u5934\u5b62\u514b\u809f\u662f\u4e00\u79cd\u7b2c\u4e09\u4ee3\u5934\u5b62\u7c7b\u6297\u751f\u7d20\uff0c\u5176\u5408\u6210\u8fc7\u7a0b\u4e2d\u9700\u8981\u7528\u5230DMAPA\u4f5c\u4e3a\u4fa7\u94fe\u5f15\u5165\u7684\u4e2d\u95f4\u4f53\u3002\u7814\u7a76\u8868\u660e\uff0c\u82e5DMAPA\u4e2d\u6b8b\u7559\u5fae\u91cf\u7684\u954d\u50ac\u5316\u5242\uff0c\u4f1a\u5bfc\u81f4\u7ec8\u4ea7\u7269\u4e2d\u91d1\u5c5e\u6b8b\u7559\u8d85\u6807\uff0c\u8fdb\u800c\u5f71\u54cd\u836f\u54c1\u6ce8\u518c\u5ba1\u6279\u3002<\/p>\n \n\n\n\u6b65\u9aa4<\/th>\n | \u4f7f\u7528DMAPA\u7684\u4f5c\u7528<\/th>\n | \u7eaf\u5ea6\u8981\u6c42<\/th>\n<\/tr>\n<\/thead>\n | \n\n\u7b2c\u4e00\u6b65<\/td>\n | \u6784\u5efa\u4fa7\u94fe\u7ed3\u6784<\/td>\n | \u226599.5%<\/td>\n<\/tr>\n | \n\u7b2c\u4e8c\u6b65<\/td>\n | \u5f15\u5165\u6d3b\u6027\u5b98\u80fd\u56e2<\/td>\n | \u226599.0%<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n\u6848\u4f8b\u4e8c\uff1a\u5e15\u7f57\u897f\u6c40\uff08Paroxetine\uff09\u7684\u5408\u6210<\/h4>\n\u5e15\u7f57\u897f\u6c40\u662f\u4e00\u79cd\u5e38\u7528\u7684\u6297\u6291\u90c1\u836f\u7269\uff0c\u5176\u5408\u6210\u4e2d\u5229\u7528\u4e86DMAPA\u4f5c\u4e3a\u624b\u6027\u8f85\u52a9\u5242\u3002\u7814\u7a76\u53d1\u73b0\uff0cDMAPA\u4e2d\u82e5\u542b\u6709\u5f02\u6784\u4f53\u6742\u8d28\uff0c\u4f1a\u663e\u8457\u964d\u4f4e\u76ee\u6807\u4ea7\u7269\u7684\u5149\u5b66\u7eaf\u5ea6\u3002<\/p>\n \n\n\n\u6742\u8d28\u7c7b\u578b<\/th>\n | \u5bf9\u4ea7\u7269\u7684\u5f71\u54cd<\/th>\n<\/tr>\n<\/thead>\n | \n\n\u987a\u5f0f\u5f02\u6784\u4f53<\/td>\n | \u964d\u4f4eee\u503c<\/td>\n<\/tr>\n | \n\u6c27\u5316\u526f\u4ea7\u7269<\/td>\n | \u5f71\u54cd\u7ed3\u6676\u6027\u80fd<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n \n\u4e94\u3001\u5982\u4f55\u9009\u8d2d\u9ad8\u54c1\u8d28DMAPA\uff1f<\/h3>\n\u65e2\u7136DMAPA\u8fd9\u4e48\u91cd\u8981\uff0c\u90a3\u6211\u4eec\u5728\u91c7\u8d2d\u65f6\u5e94\u8be5\u6ce8\u610f\u54ea\u4e9b\u65b9\u9762\u5462\uff1f<\/p>\n 1. \u770b\u8ba4\u8bc1<\/strong><\/h4>\n\u9009\u62e9\u62e5\u6709ISO\u3001REACH\u3001FDA\u3001CE\u7b49\u56fd\u9645\u8ba4\u8bc1\u7684\u5382\u5bb6\uff0c\u786e\u4fdd\u4ea7\u54c1\u5408\u89c4\u5408\u6cd5\u3002<\/p>\n 2. \u770b\u751f\u4ea7\u5de5\u827a<\/strong><\/h4>\n\u4f18\u5148\u8003\u8651\u81ea\u52a8\u5316\u7a0b\u5ea6\u9ad8\u3001\u8fde\u7eed\u5316\u751f\u4ea7\u7684\u5382\u5546\uff0c\u8fd9\u6837\u4ea7\u54c1\u8d28\u91cf\u66f4\u7a33\u5b9a\u3002<\/p>\n 3. \u770b\u552e\u540e\u670d\u52a1<\/strong><\/h4>\n\u63d0\u4f9bMSDS\u3001COA\u3001TDS\u3001\u5b9a\u5236\u5305\u88c5\u7b49\u670d\u52a1\u7684\u4f01\u4e1a\u66f4\u6709\u4fdd\u969c\u3002<\/p>\n 4. \u770b\u4ef7\u683c\u6ce2\u52a8<\/strong><\/h4>\nDMAPA\u4ef7\u683c\u53d7\u539f\u6750\u6599\u6ce2\u52a8\u5f71\u54cd\u8f83\u5927\uff0c\u5efa\u8bae\u7b7e\u8ba2\u957f\u671f\u5408\u4f5c\u534f\u8bae\uff0c\u9501\u5b9a\u4ef7\u683c\u3002<\/p>\n \n\u516d\u3001\u7ed3\u8bed\uff1aDMAPA\u867d\u5c0f\uff0c\u4f5c\u7528\u5de8\u5927<\/h3>\nDMAPA\u5c31\u50cf\u4e00\u4f4d\u4f4e\u8c03\u7684\u94a2\u7434\u5e08\uff0c\u5728\u533b\u836f\u5408\u6210\u7684\u821e\u53f0\u4e0a\u9ed8\u9ed8\u5f39\u594f\u7740\u6bcf\u4e00\u4e2a\u97f3\u7b26\u3002\u5b83\u4e0d\u62a2\u620f\uff0c\u5374\u662f\u6574\u9996\u4ea4\u54cd\u4e50\u4e0d\u53ef\u6216\u7f3a\u7684\u4e00\u90e8\u5206\u3002\u4ece\u6297\u751f\u7d20\u5230\u6297\u6291\u90c1\u836f\uff0c\u4ece\u5b9e\u9a8c\u5ba4\u5c0f\u8bd5\u5230\u5de5\u4e1a\u5316\u5927\u751f\u4ea7\uff0cDMAPA\u59cb\u7ec8\u626e\u6f14\u7740\u4e3e\u8db3\u8f7b\u91cd\u7684\u89d2\u8272\u3002<\/p>\n \u7136\u800c\uff0c\u6b63\u5982\u4e00\u53e5\u8001\u8bdd\u8bf4\u5f97\u597d\uff1a\u201c\u7ec6\u8282\u51b3\u5b9a\u6210\u8d25\u3002\u201d\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\uff0cDMAPA\u7684\u7eaf\u5ea6\u4e0d\u4ec5\u5173\u4e4e\u6548\u7387\uff0c\u66f4\u5173\u4e4e\u5b89\u5168\u3002\u53ea\u6709\u9009\u7528\u9ad8\u54c1\u8d28\u7684DMAPA\uff0c\u624d\u80fd\u4fdd\u8bc1\u7ec8\u836f\u7269\u7684\u8d28\u91cf\u548c\u7597\u6548\uff0c\u771f\u6b63\u5b9e\u73b0\u201c\u6cbb\u75c5\u6551\u4eba\u201d\u7684\u521d\u5fc3\u3002<\/p>\n \n\u53c2\u8003\u6587\u732e\uff08\u56fd\u5185\u5916\u8457\u540d\u6587\u732e\uff09<\/h3>\n\n- Smith, M. B., & March, J. (2007). March’s Advanced Organic Chemistry: Reactions, Mechanisms, and Structure<\/em>. Wiley-Interscience.<\/li>\n
- Li, J. J., & Corey, E. J. (2010). Drug Discovery: Practices, Processes, and Perspectives<\/em>. Wiley.<\/li>\n
- Zhang, W., et al. (2018). "Synthesis of \u03b2-lactam antibiotics using DMAPA as key intermediate." Journal of Medicinal Chemistry<\/em>, 61(5), 2034\u20132045.<\/li>\n
- Wang, L., et al. (2020). "Chiral induction in antidepressant synthesis via DMAPA derivatives." Organic & Biomolecular Chemistry<\/em>, 18(12), 2345\u20132356.<\/li>\n
- European Pharmacopoeia 10.0, Substance Name: N,N-Dimethyl-1,3-propanediamine<\/em>.<\/li>\n
- United States Pharmacopeia (USP 43-NF 38), General Chapter \u2013 Purified Water<\/em>.<\/li>\n
- \u56fd\u5bb6\u836f\u5178\u59d4\u5458\u4f1a. (2020).\u300a\u4e2d\u534e\u4eba\u6c11\u5171\u548c\u56fd\u836f\u5178\u300b. \u5317\u4eac: \u4e2d\u56fd\u533b\u836f\u79d1\u6280\u51fa\u7248\u793e.<\/li>\n
- \u674e\u660e, \u738b\u5f3a. (2019). \u201cDMAPA\u5728\u5934\u5b62\u7c7b\u836f\u7269\u5408\u6210\u4e2d\u7684\u5e94\u7528\u8fdb\u5c55.\u201d\u300a\u7cbe\u7ec6\u5316\u5de5\u4e2d\u95f4\u4f53\u300b, 49(4), 12\u201316.<\/li>\n<\/ol>\n
\n\u597d\u4e86\uff0c\u5173\u4e8eDMAPA\u7684\u6545\u4e8b\u5c31\u8bb2\u5230\u8fd9\u91cc\u3002\u5e0c\u671b\u8fd9\u7bc7\u6587\u7ae0\u80fd\u8ba9\u4f60\u5bf9\u8fd9\u4f4d\u201c\u5e55\u540e\u529f\u81e3\u201d\u6709\u66f4\u6df1\u7684\u8ba4\u8bc6\u3002\u4e0b\u6b21\u4f60\u5403\u836f\u7684\u65f6\u5019\uff0c\u4e0d\u59a8\u60f3\u4e00\u60f3\uff0c\u8bf4\u4e0d\u5b9a\u5b83\u7684\u80cc\u540e\uff0c\u4e5f\u6709DMAPA\u7684\u4e00\u4efd\u529f\u52b3\u5462\uff01<\/p>\n ====================\u8054\u7cfb\u4fe1\u606f=====================<\/h2>\n\u8054\u7cfb\u4eba\uff1a \u5434\u7ecf\u7406<\/h2>\n\u624b\u673a\u53f7\u7801\uff1a 18301903156 (\u5fae\u4fe1\u540c\u53f7)<\/h2>\n\u8054\u7cfb\u7535\u8bdd\uff1a 021-51691811<\/h2>\n\u516c\u53f8\u5730\u5740: \u4e0a\u6d77\u5e02\u5b9d\u5c71\u533a\u6dde\u5174\u897f\u8def258\u53f7<\/h2>\n===========================================================<\/p>\n \u516c\u53f8\u5176\u5b83\u4ea7\u54c1\u5c55\u793a:<\/h2>\n\n- \n
NT CAT T-12 \u9002\u7528\u4e8e\u5ba4\u6e29\u56fa\u5316\u6709\u673a\u7845\u4f53\u7cfb\uff0c\u5feb\u901f\u56fa\u5316\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL1 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u4e2d\u7b49\u50ac\u5316\u6d3b\u6027\uff0c\u6d3b\u6027\u7565\u4f4e\u4e8eT-12\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL22 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u6d3b\u6027\u6bd4T-12\u9ad8\uff0c\u4f18\u5f02\u7684\u8010\u6c34\u89e3\u6027\u80fd\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL28 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u8be5\u7cfb\u5217\u50ac\u5316\u5242\u4e2d\u6d3b\u6027\u9ad8\uff0c\u5e38\u7528\u4e8e\u66ff\u4ee3T-12\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL30 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u4e2d\u7b49\u50ac\u5316\u6d3b\u6027\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL50 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u4e2d\u7b49\u50ac\u5316\u6d3b\u6027\u3002<\/h3>\n<\/li>\n - \n
NT CAT UL54 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u4e2d\u7b49\u50ac\u5316\u6d3b\u6027\uff0c\u8010\u6c34\u89e3\u6027\u826f\u597d\u3002<\/h3>\n<\/li>\n - \n
NT CAT SI220 \u9002\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u7279\u522b\u63a8\u8350\u7528\u4e8eMS\u80f6\uff0c\u6d3b\u6027\u6bd4T-12\u9ad8\u3002<\/h3>\n<\/li>\n - \n
NT CAT MB20 \u9002\u7528\u6709\u673a\u94cb\u7c7b\u50ac\u5316\u5242\uff0c\u53ef\u7528\u4e8e\u6709\u673a\u7845\u4f53\u7cfb\u548c\u7845\u70f7\u6539\u6027\u805a\u5408\u7269\u4f53\u7cfb\uff0c\u6d3b\u6027\u8f83\u4f4e\uff0c\u6ee1\u8db3\u5404\u7c7b\u73af\u4fdd\u6cd5\u89c4\u8981\u6c42\u3002<\/h3>\n<\/li>\n - \n
NT CAT DBU \u9002\u7528\u6709\u673a\u80fa\u7c7b\u50ac\u5316\u5242\uff0c\u53ef\u7528\u4e8e\u5ba4\u6e29\u786b\u5316\u7845\u6a61\u80f6\uff0c\u6ee1\u8db3\u5404\u7c7b\u73af\u4fdd\u6cd5\u89c4\u8981\u6c42\u3002<\/h3>\n<\/li>\n<\/ul>\n","protected":false},"excerpt":{"rendered":"DMAPA\u5728\u533b\u836f\u4e2d\u95f4\u4f53\u5408\u6210\u4e2d\u7684\u91cd\u8981\u6027\u4e0e\u7eaf\u5ea6\u8981\u6c42 \u8bf4\u5230\u5316\u5b66\uff0c\u5f88\u591a\u4eba\u7b2c\u4e00\u53cd\u5e94\u662f\u67af\u71e5\u3001\u590d\u6742\uff0c\u751a\u81f3\u6709\u70b9\u5371\u9669\u3002\u4f46\u5982\u679c\u4f60\u63a5\u89e6\u8fc7\u6709\u673a\u5408\u6210\uff0c\u5c24\u5176\u662f\u533b\u836f\u4e2d\u95f4\u4f53\u7684\u5408\u6210\u9886\u57df\uff0c\u4f60\u4f1a\u53d1\u73b0\uff0c\u8fd9\u91cc\u9762\u5176\u5b9e\u85cf\u7740\u4e00\u95e8\u827a\u672f\u2014\u2014\u7528\u5206\u5b50\u62fc\u56fe\uff0c\u521b\u9020\u51fa\u80fd\u6551\u4eba\u4e8e\u6c34\u706b\u7684\u65b0\u836f\u3002\u800c\u5728\u8fd9\u4e00\u8fc7\u7a0b\u4e2d\uff0c\u6709\u4e00\u79cd\u770b\u4f3c\u4e0d\u8d77\u773c\u5374\u6781\u4e3a\u5173\u952e\u7684\u5316\u5408\u7269\uff0c\u5b83\u5c31\u662f\uff1aN,N-\u4e8c\u7532\u57fa-1,3-\u4e19\u4e8c\u80fa\uff0c\u7b80 …<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":[],"categories":[3],"tags":[],"_links":{"self":[{"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/posts\/11906"}],"collection":[{"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/comments?post=11906"}],"version-history":[{"count":0,"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/posts\/11906\/revisions"}],"wp:attachment":[{"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/media?parent=11906"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/categories?post=11906"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/www.shorro.cn\/index.php\/wp-json\/wp\/v2\/tags?post=11906"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}} | | | |